Phomopsidin
WebThis manuscript describes an alternative synthetic approach for (+)-phomopsidin, which shows strong inhibitory activity against the assembly of microtubule proteins. We observed that the TADA reaction of the macrolactone 5 with the reversed C11 configuration provided the desired cycloadduct 6 in 86% yield with excellent stereoselectivity (dr=16:1).
Phomopsidin
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WebHis research there focused on the use of the Diels-Alder reaction and intramolecular rearrangements (specifically lactonic Ireland-Claisen rearrangements) to rapidly synthesize the marine natural products Phomopsidin and Aspermytin A. He is a natural product/total synthesis organic chemist at heart. WebJan 20, 2003 · Phomopsidin and its (16Z)-isomer (MK8383) showed anti-microtubule activity at IC 50 of 5.7 and 8.0 μM, respectively, while the Me ester and other compounds were not active at 100 μM. The absolute configuration of phomopsidin ( 1 ) was …
Webphosphamidon: [noun] a contact and systemic organophosphorus insecticide and miticide C10H19ClNO5P. WebDec 5, 2012 · The Journal of Antibiotics - Identification of a new phomoxanthone antibiotic from Phomopsis longicolla and its antimicrobial correlation with other metabolites during fermentation
WebAbstract The absolute configuration of phomopsidin, a marine-derived fungal metabolite from Phomopsis sp. isolated at Pohnpei, was determined by the exciton chirality method as 6S, 7S, 8S, 11S, 12R, and 15R. The biosynthetic study using 13C-labeled precursors revealed the origin of all carbon atoms in phomopsidin, which was built by nine acetates and three … WebPhomopsidin. Catalog No. T125428 CAS 199173-60-9. All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use. Phomopsidin, CAS 199173-60-9 Please contact us for prices and availability for the specification of product you are interested at. Product consultation. Get quote ...
WebJan 24, 2009 · In 1997, (+)-phomopsidin ( Fig. 1) was isolated from a marine-derived fungus, Phomopsis sp. strain TUF 95F47, that was collected in Pohnpei. 1 (+)-Phomopsidin was …
WebJun 29, 2004 · Read "First Total Synthesis of Antimitotic Compound, (+)‐Phomopsidin., ChemInform" on DeepDyve, the largest online rental service for scholarly research with thousands of academic publications available at your fingertips. fob food mapWebApr 24, 2024 · During a survey of xylarialean fungi in Northern Iran, several specimens that showed affinities to the Hypoxylon rubiginosum complex were collected and cultured. A comparison of their morphological characters, combined with a chemotaxonomic study based on high performance liquid chromatography, coupled with diode array detection … greeny sports showWebDec 5, 2012 · The Journal of Antibiotics - Identification of a new phomoxanthone antibiotic from Phomopsis longicolla and its antimicrobial correlation with other metabolites during … greeny suhrWebJan 24, 2009 · In 1997, (+)-phomopsidin ( Fig. 1) was isolated from a marine-derived fungus, Phomopsis sp. strain TUF 95F47, that was collected in Pohnpei. 1 (+)-Phomopsidin was found to be a new inhibitor of microtubule assembly, showing strong inhibitory activity against the assembly of microtubule proteins derived from the porcine brain at an IC 50 of … greeny show staffWebAbstract. (Equation presented) The first total synthesis of (+)-phomopsidin has been achieved via a diastereoselective transannular Diels-Alder (TADA) reaction. Key steps in … fob fas 違いWebMK8383, isolated from Phoma sp. T2526 in 1993, exhibits potent antibiotic activities against a variety of phytopathogens and has been considered a promising fungicide against Botrytis cinerea. Unfortunately, MK8383 is a photosensitive compound and it … greenys taxis seahamWebPhomopsidin, a new inhibitor of microtubule assembly produced by Phomopsis sp. isolated from coral reef in Pohnpei J Antibiot (Tokyo). 1997 Oct;50 (10):890-2. doi: … fob for car meaning